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| Item No | Product Name | Product Description | Product Description | Inquiry |
|---|---|---|---|---|
| R-SX-383 | MPEP hydrochloride,CAS219911-35-0 | MPEP is a potent, highly selective non-competitive antagonist at the mGlu5a receptor subtype (IC50 = 36 nM) while having no agonist or antagonist activities at the mGlu1b receptor at concentrations up to 30 uM.西安瑞禧生物提供各種抑制劑材料。 | 查看詳細(xì) | |
| R-SX-384 | TG6-10-1,CAS1415716-58-3 | TG6-10-1 是一種 EP2 拮抗劑, 低納摩爾下有效作用于 EP2, 比作用于人 EP3, EP4 和 IP 受體選擇性高 300, EP1 受體選擇性高 100 倍的。西安瑞禧生物提供各種抑制劑材料。 | 查看詳細(xì) | |
| R-SX-385 | Elacridar HCl,CAS143851-98-3 | Elacridar hydrochloride is a P-glycoprotein inhibitor, and has been used both in vitro and in vivo as a tool inhibitor of P-glycoprotein (Pgp) to investigate the role of transporters in the disposition of various test molecules.西安瑞禧生物提供各種抑制劑材料。 | 查看詳細(xì) | |
| R-SX-386 | Muscimol HBr,CAS18174-72-6 | Muscimol hydrobromide is a potent but toxic structural analog of g-aminobutyric acid (GABA), with a zwitterionic structure西安瑞禧生物提供各種抑制劑材料。 | 查看詳細(xì) | |
| R-SX-388 | MK-801 ; Dizocilpine,CAS77086-21-6 | MK-801 (Dizocilpine) is a potent N-methyl-D-aspartate (NMDA) receptor antagonist with Ki of 30.5 nM.西安瑞禧生物提供各種抑制劑材料。 | 查看詳細(xì) | |
| R-SX-389 | Iloperidone,CAS133454-47-4 | Iloperidone(HP 873)是D2/5-HT2受體拮抗劑，可作用于精神分裂癥。西安瑞禧生物提供各種抑制劑材料。 | 查看詳細(xì) | |
| R-SX-390 | Bromfenac sodium,CAS91714-93-1 | Bromfenac Sodium是一種非甾體類抗炎藥(NSAID)，具有抗炎活性，通過抑制環(huán)氧合酶1和2可阻斷前列腺素的合成。西安瑞禧生物提供各種抑制劑材料。 | 查看詳細(xì) | |
| R-SX-391 | VU0361737,CAS1161205-04-4 | VU 0361737 is a selective positive allosteric modulator (PAM) for mGlu4 receptor with EC50 of 240 nM and 110 nM at human and rat receptors, respectively, displays weak activity at mGlu5 and mGlu8 receptors, is inactive at mGlu1, mGlu2, mGlu3, mGlu6 and mGlu7 receptors, can penetrate into CNS.西安瑞禧生物提供各種抑制劑材料。 | 查看詳細(xì) | |
| R-SX-392 | VU0357121,CAS433967-28-3 | VU0357121 is a novel positive allosteric modulator (PAM) of mGlu5 with EC50 of 33 nM, is inactive or very weakly antagonizing at other mGlu receptor subtypes.西安瑞禧生物提供各種抑制劑材料。 | 查看詳細(xì) | |
| R-SX-393 | VU0364770,CAS61350-00-3 | VU 0364770 is a positive allosteric modulator(PAM) of mGlu4 with EC50 of 1.1 μM, exhibits insignificant activity at 68 other receptors, including other mGlu subtypes.西安瑞禧生物提供各種抑制劑材料。 | 查看詳細(xì) | |
| R-SX-394 | Ivabradine hydrochloride,CAS148849-67-6 | Ivabradine hydrochloride 是可口服的，超極化激活的環(huán)核苷酸門控離子通道 (HCN) 通道阻滯劑。西安瑞禧生物提供各種抑制劑材料。 | 查看詳細(xì) | |
| R-SX-395 | BRL54443,CAS57477-39-1 | BRL 54443是5-HT1E/1F受體激動劑，pKi分別為8.7和8.9，比對其它5-HT和多巴胺受體的抑制性高30倍以上。西安瑞禧生物提供各種抑制劑材料。 | 查看詳細(xì) | |
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